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Testosterone Cypionate

Also sold as Test Cyp, Depo-Testosterone.

Half-life
190 h
Steady state
~40 d
Class
Androgen
Category
TRT

Published population averages. Steady state is the usual five half-life rule of thumb, not a measurement. See peptide half-life, explained.

Overview

Testosterone Cypionate is the most commonly prescribed testosterone ester in the United States for testosterone replacement therapy (TRT). It is a long-acting intramuscular injectable that provides stable testosterone levels with weekly or biweekly dosing. It is essentially identical to Testosterone Enanthate with a marginally longer half-life.

How it works

After intramuscular injection, the cyclopentylpropionic acid ester is cleaved by tissue esterases, releasing free testosterone. Testosterone then binds androgen receptors (AR) in target tissues, and is also converted to dihydrotestosterone (5α-reductase) and estradiol (aromatase) for additional effects. Suppresses gonadotropins (LH, FSH) via hypothalamic feedback.

Half-life and peak

Terminal half-life approximately 8 days (~190 hours). Peak serum levels reached 24–48 hours post-IM injection. Nadir occurs around day 7, supporting weekly dosing. Subcutaneous injection shows similar PK with slightly lower Cmax.

What it is studied for

Male hypogonadism, TRT optimization, cardiovascular safety (TRAVERSE trial), bone mineral density, body composition, sexual function, mood and cognition.

Research status

FDA-approved (Depo-Testosterone). TRAVERSE cardiovascular safety trial (2023, NEJM) established non-inferiority to placebo for MACE in men with hypogonadism. Decades of clinical experience.

Sources

Educational reference only. This page describes what is published about a compound; it is not medical advice, not a recommendation to take anything, and not a dosing guide. Several compounds in this catalog are investigational and are not approved medicines. Talk to a doctor.

Guides that cover it